2015年1月12日 星期一

Pharmaceutical Intermediates

Name of APIName Of IntermediateCAS#
Abiraterone 3-Diethylboranyl Pyridine89878-14-8
Abiraterone 3-Pyridyl bromide626-55-1
Abiraterone17-Iodoandrosta-5,16-dien-3beta-ol32138-69-5
Abirateronetert-Butyl (4R,6R)-2-[[[6-(2-4-fluorophenyl)-5-isopropyl-3-phenyl-4-(phenylcarbamoyl)pyrrol-1-yl]ethyl]-2,2-dimethyl-1,3-dioxan-4-yl]acetate125971-95-1
Abiraterone4-Fluoro-alpha-(2-methyl-1-oxopropyl)-gamma-oxo-N,bata-diphenylbenzene butaneamide125971-96-2
Bosentan hydrate Diethyl Bromoalonate685-87-0
Canagliflozin 2-(5-bromo-2-methylbenzyl)-5-(4-fluorophenyl)thiophene 1030825-20-7
Canagliflozin 2-(4-Fluorophenyl)thiophene 58861-48-6
Canagliflozin (3R,4S,5R,6R)-3,4,5-tris(triMethylsilyloxy)-6-((triMethylsilyloxy)Methyl)tetrahydro-2H-pyran-2-one32384-65-9
Canagliflozin (5-(4-Fluorophenyl)thiophen-2-yl)(5-iodo-2-methylphenyl)methanone1071929-08-2
Canagliflozin (5-bromo-2-methylphenyl)(5-(4-fluorophenyl)thiophen-2-yl)methanone1132832-75-7
Cyclopropylboronic acidBromocyclopropane4333-56-6
Dofetilide N-Methyl-4-nitrophenethylamine hydrochloride166943-39-1
Dofetilide 1-(2-Chloroethoxy)-4-nitrobenzene3383-72-0
Esomeprazole Sodium3,5-Dimethyl-4-methoxy-2-pyridinemethanol86604-78-6
Esomeprazole Sodium 5-Methoxy-2-mercaptobenzimidazole37052-78-1
Etravirine3,5-Dimethyl-4-hydroxybenzaldehyde2233-18-3
Etravirine4-Aminobenzonitrile873-74-5
Etravirine 4-(4,6-dichloropyrimidin-2-ylamino)benzonitrile329187-59-9
Etravirine 4-((5-bromo-4,6-dichloro-2-pyrimidinyl)amino)benzonitrile269055-75-6
Etravirine  4-((5-bromo-6-chloro-2-((4-cyanophenyl)amino)-4-pyrimidinyl)oxy)-3,5-dimethylbenzonitrile269055-76-7
Fulvestrant  9-Bromo-1-nonanol55362-80-6
Lurasidone3-(1-Piperazinyl)-1,2-benzisothiazole87691-87-0
Lurasidone(1R,2R)-1,2-Cyclohexanedimethanol65376-05-8
Lurasidone(1R,2R)-1,2-Cyclohexanedicarboxylic acid46022-05-3
Lurasidone(3aR,4S,7R,7aS)-hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione14805-29-9
Oxaliplatin(1R,2R)-(-)-1,2-Diaminocyclohexane20439-47-8
Praziquantel2-(Phenylcarbonyl)-1,2,3,6,7,11b-hexahydro-4H-pyrazino[2,1-a]isoquinolin-4-one54761-87-4
Silodosin2-[2-(2,2,2-Trifluoroethoxy)phenoxy]ethyl methanesulfonate160969-03-9
Silodosin2-(2,2,2-Trifluoroethoxy)phenol160968-99-0
Silodosin2-[2-(2,2,2-Trifluoroethoxy)phenoxy]-ethyl bromide 160969-00-6
Silodosin5-[(2R)-2-Aminopropyl]-1-[3-(benzoyloxy)propyl]-2,3-dihydro-1H-indole-7-carbonitrile (2R,3R)-2,3-dihydroxybutanedioate 239463-85-5
Esomeprazole 4-Methoxy-3,5-dimethyl-2-pyridinemethanol86604-78-6
Ufiprazole2-{[(3,5-Dimethyl-4-methoxy-2-pyridinyl)-methyl]-thio}-5-methoxy-1H-benzimidazole73590-85-9
Tolvaptano-Toluoyl chloride933-88-0
Tolvaptan2-Methyl-4-nitrobenzoic acid1975-51-5
Tolvaptan7-Chloro-1,2,3,4-tetrahydrobenzo[b]azepin-5-one160129-45-3
ErlotinibEthyl 4,5-bis(2-methoxyethoxy)-2-aminobenzoate179688-27-8
Erlotinib3-Aminophenylacetylene54060-30-9
Ambrisentan4,6-Dimethyl-2-(methylsulfonyl)pyrimidine35144-22-0
Vilazodone 1-Boc-piperazine57260-71-6
Vilazodone Indole-5-carbonitrile15861-24-2
Vilazodone Ethyl 5-bromobenzofuran-2-carboxylate84102-69-2
Rasagiline          Propargyl Benzenesulfonate6165-75-9
Rasagiline         Propargyl p-toluenesulfonate6165-76-0
Rasagiline          (R)-(-)-1-Aminoindan10277-74-4
Rasagiline            Rasagiline136236-51-6
Rilpivirine                  4-Iodo-2,6-dimethylaniline4102-53-8
Rilpivirine                    4-[(4-Chloro-2-pyrimidinyl)amino]benzonitrile244768-32-9
Roflumilast4-Amino-3,5-dichloropyridine22889-78-7 
Roflumilast 3-(Cyclopropylmethoxy)-4-hydroxybenzoic acid1243391-44-7
Rosuvastatin        Dimethyl-3-Hydroxyglutarate7250-55-7
Rosuvastatin         Diethyl-3-Hydroxyglutarate32328-03-3
Rosuvastatin            Methyl (3R)-3-(tert-butyldimethylsilyloxy)-5-oxo-6-triphenylphosphoranylidenehexanoate147118-35-2
Saxagliptin Hcl         (1S,3S,5S)-tert-butyl 3-carbamoyl-2-aza-bicyclo[3.1.0]hexane-2-carboxylate361440-67-7
Saxagliptin Hcl        (S)-1-tert-butyl 2-ethyl 2,3-dihydropyrrole-1,2-dicarboxylate178172-26-4
Saxagliptin Hcl           (S)-1-tert-butyl 2-ethyl 5-oxopyrrolidine-1,2-dicarboxylate144978-12-1
Saxagliptin Hcl            (S)-tert-butyl 2-carbamoyl-2,3-dihydropyrrole-1-carboxylate709031-38-9
Strontium Diethyl 1,3-acetone Dicarboxylate105-50-0
Strontium Ethyl 5-amino-4-cyano-3-(2-ethoxy-2-oxoethyl)thiophene-2-carboxylate58168-20-0
Strontium Tetraethyl ranelate58194-26-6
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